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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50316887'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  6.5nMAssay Description:Antagonist activity at human recombinant adenosine receptor A2a by cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  6.5nMAssay Description:Antagonistic activity at adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  6.5nMAssay Description:Antagonist activity at human Adenosine receptor A2a assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50316887(2-amino-8-(2-morpholinoethoxy)-4-phenyl-5H-indeno[...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]MSX-2 from human recombinant adenosine A2A receptor expressed in CHO cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed