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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50339077'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50339077((2R,3R,4S)-2-(6-amino-2-((E)-hex-1-enyl)-9H-purin-...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50339077((2R,3R,4S)-2-(6-amino-2-((E)-hex-1-enyl)-9H-purin-...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50339077((2R,3R,4S)-2-(6-amino-2-((E)-hex-1-enyl)-9H-purin-...)
Affinity DataEC50:  20.6nMAssay Description:Agonist activity at human recombinant adenosine A2A receptor expressed in CHO cells assessed as induction of cAMP production after 30 mins by immunoa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed