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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM21217'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Napoli

LigandPNGBDBM21217(2-(4-methyl-1H-1,3-benzodiazol-2-yl)quinoxaline | ...)
Affinity DataKi:  26nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A3 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Napoli

LigandPNGBDBM21217(2-(4-methyl-1H-1,3-benzodiazol-2-yl)quinoxaline | ...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]I-AB-MECA from human recombinant adenosine A3 receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universita Di Napoli

LigandPNGBDBM21217(2-(4-methyl-1H-1,3-benzodiazol-2-yl)quinoxaline | ...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed