Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50051361'
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50051361(3-Methylsulfanyl-6,7-dihydro-benzo[c]thiophene-1-c...)
Affinity DataKi:  1.30E+4nMAssay Description:Binding affinity against human adenosine A3 receptor in HEK293 cells using [125I]-AB-MECA 21680 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50051361(3-Methylsulfanyl-6,7-dihydro-benzo[c]thiophene-1-c...)
Affinity DataKi:  1.31E+4nMAssay Description:Displacement of [125I]-AB-MECA from rat Adenosine A3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed