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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50109488'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50109488(4-(3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-MRE3008-F20 from human Adenosine A3 receptor expressed in HEK cells; range 31-50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50109488(4-(3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  40nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50109488(4-(3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50109488(4-(3-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed