Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50125911'
TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50125911(1-(9-Ethylamino-2-furan-2-yl-8-methyl-8H-pyrazolo[...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]- MRE 308F20 binding from human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125911(1-(9-Ethylamino-2-furan-2-yl-8-methyl-8H-pyrazolo[...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]- MRE 308F20 binding from human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50125911(1-(9-Ethylamino-2-furan-2-yl-8-methyl-8H-pyrazolo[...)
Affinity DataIC50:  45nMAssay Description:Antagonist activity as inhibition of cAMP generation after agonist-modulation of Adenosine A3 receptor with 100 nM CI-IB-MECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed