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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50185937'
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50185937(3-azido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydr...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor H272D mutant expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50185937(3-azido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydr...)
Affinity DataKi:  186nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor H272E mutant expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50185937(3-azido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydr...)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor T94A mutant expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50185937(3-azido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydr...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [125I]I-AB-MECA from human adenosine A3 receptor T94E mutant expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50185937(3-azido-5-(6-(3-iodobenzylamino)purin-9-yl)-4-hydr...)
Affinity DataKi:  2.26E+3nMAssay Description:Displacement of [125I]I-AB-MECA from wild type adenosine A3 receptor expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed