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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50245931'
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245931(5-methyl-N-(2-phenyl-2H-pyrazolo[3,4-c]quinolin-4-...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50245931(5-methyl-N-(2-phenyl-2H-pyrazolo[3,4-c]quinolin-4-...)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as inhibition of CI-IB-MECA-mediated inhibition of cAMP accumulati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed