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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50300684'
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50300684(5-methyl-2-p-tolyl-2H-pyrazolo[4,3-d]pyrimidin-7(6...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]AB-MECA from human cloned adenosine A3 receptor expressed in CHO cells after 120 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50300684(5-methyl-2-p-tolyl-2H-pyrazolo[4,3-d]pyrimidin-7(6...)
Affinity DataKi:  46nMAssay Description:Antagonist activity at human cloned adenosine A3 receptor expressed in CHO cells assessed as inhibition of Cl-IB-MECA-inhibited [3H]cAMP production b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed