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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50318269'
TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50318269(1-(2-benzyl-6-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50318269(1-(2-benzyl-6-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4...)
Affinity DataIC50:  8.20nMAssay Description:Antagonist activity human recombinant adenosine A3 receptor expressed in CHO cells assessed as blockade of NECA-mediated inhibition of forskolin-stim...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed