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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50379127'
TargetAdenosine receptor A3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379127(CHEMBL2012672)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]AB-MECA from human recombinant adenosine receptor-3 expressed in CHO cell membrane after 60 mins by gamma-countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379127(CHEMBL2012672)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]I-AB-MECA from human A3 adenosine receptor expressed in CHO cells after 60 min Packard Cobra 2 gamma-counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed