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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50389899'
TargetAdenosine receptor A3(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50389899(CHEMBL2070882)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]MRE-3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50389899(CHEMBL2070882)
Affinity DataIC50:  301nMAssay Description:Antagonist activity at human adenosine A3 receptor expressed in CHO cells assessed as forskolin/C1-IB-MECA-induced inhibition of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed