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Found 12 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM85619'
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [125]AB-MECA from human Adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells; range 0.85-0.98More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.910nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]-MRE3008-F20 binding at human Adenosine A3 receptor expressed in HEK cells; range 0.85-0.98More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.910nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.910nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.910nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.980nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataIC50:  5.30nMAssay Description:Inhibitory concentration as antagonistic activity against cAMP generation inhibited by IB-MECA in CHO cell membranes transfected with human A3 recept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Ferrara

Curated by PDSP Ki Database
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of cAMP accumulation in CHO cells expressing human adenosine A3 receptor; range 4.0-7.5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed