TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]prazosin from human adrenergic alpha1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]prazosin from human recombinant alpha1A adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.0700nMAssay Description:Inhibition of [3H]- prazosin binding against Alpha-1A adrenergic receptor from rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.126nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]prazosin from alpha1-adrenoceptor (unknown origin) in cerebral cortex membranes after 60 mins by TopCount scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Binding affinity against Alpha-1A adrenergic receptor from bovine cloneMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.230nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.270nMAssay Description:Ability to displace [3H]prazosin from cloned human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.300nMAssay Description:Compound was evaluated for its ability to displace [125I]-HEAT binding from rat Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.390nMAssay Description:Compound was tested for binding affinity utilizing cloned receptor binding assays by using [125 I]HEAT as radioligand to the human Alpha-1A adrenergi...More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Binding affinity against Alpha-1A adrenergic receptor from human cloneMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:Binding affinity against human Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.580nMAssay Description:The compound was tested for binding affinity on [3H]- prazosin as specific ligand on Human cloned alpha-1A adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.588nMAssay Description:Binding affinity to adrenergic alpha1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.589nMAssay Description:Binding affinity measured in CHO cells expressing human cloned Alpha-1A adrenergic receptor expressed as pKiMore data for this Ligand-Target Pair
Affinity DataKi: 0.589nMAssay Description:Displacement of [3H]prazosin from human alpha1A adrenoceptor expressed in CHO cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.589nMAssay Description:Binding affinity to adrenergic alpha1A receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding affinity against alpha-1A adrenergic receptor of human liver microsomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.610nMAssay Description:Binding affinity towards human cloned alpha1A-adrenoceptor using [3H]-prazosin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.724nMAssay Description:Compound was tested for binding affinity against cloned Alpha-1A adrenergic receptor from bovine brain using radioligand ([3H]prazosin) binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.930nMAssay Description:Displacement of [3H]prazosin (0.3 nM) from bovine Alpha-1A adrenergic receptor expressed in BHK cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 0.933nMAssay Description:Binding affinity against native Alpha-1A adrenergic receptor from rat hippocampus pretreated with chloroethylclonidine using radioligand ([3H]prazosi...More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataKi: 1.05nMAssay Description:Compound was tested for its binding affinity towards Alpha-1A adrenergic receptor using [3H]-prazosin from rat submaxillary glandMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Unwersity Of Misscuri
Curated by PDSP Ki Database
Unwersity Of Misscuri
Curated by PDSP Ki Database
Affinity DataIC50: 0.254nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1A receptor in Wistar rat submaxillary gland after 60 minsMore data for this Ligand-Target Pair