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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-1D adrenergic receptor' and Ligand = 'BDBM50418765'
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50418765(CHEMBL1796046)
Affinity DataKi:  0.501nMAssay Description:Antagonist activity against human cloned adrenergic Alpha-1D receptor expressed in HEK293 cells assessed as inhibition of norepinephrine-induced [3H]...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50418765(CHEMBL1796046)
Affinity DataKi:  14.4nMAssay Description:Displacement of [125I]BE-2254 from human adrenergic Alpha-1D receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed