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Found 5 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50030622'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50030622((7aS,8S,11aS,12aR)-8-Methyl-5,6,7a,8,11a,12,12a,13...)
Affinity DataKi:  71nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50030622((7aS,8S,11aS,12aR)-8-Methyl-5,6,7a,8,11a,12,12a,13...)
Affinity DataKi:  104nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50030622((7aS,8S,11aS,12aR)-8-Methyl-5,6,7a,8,11a,12,12a,13...)
Affinity DataKi:  106nMAssay Description:Inhibition of [3H]rauwolscine binding to CHO cells expressing the human Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50030622((7aS,8S,11aS,12aR)-8-Methyl-5,6,7a,8,11a,12,12a,13...)
Affinity DataKi:  130nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(BOVINE)
University Of Nebraska

Curated by PDSP Ki Database
LigandPNGBDBM50030622((7aS,8S,11aS,12aR)-8-Methyl-5,6,7a,8,11a,12,12a,13...)
Affinity DataKi:  1.83E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed