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Found 1 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50417010'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Pierre Fabre Research Center

Curated by ChEMBL
LigandPNGBDBM50417010(CHEMBL1255723)
Affinity DataKi:  0.138nMAssay Description:Displacement of [3H]-RX821002 from human adrenergic alpha2A receptor expressed in rat C6 cells after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed