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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-2A adrenergic receptor' and Ligand = 'BDBM50419888'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50419888(CHEMBL1956202)
Affinity DataKi:  1.02E+3nMAssay Description:Displacement of [3H]RS-79948-197 from human adrenoceptor aplha 2A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50419888(CHEMBL1956202)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human adrenoceptor aplha 2A expressed in CHO cells assessed as rate of extracellular acidification by cytosensor microphysiometri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed