Affinity DataKi: 126nMAssay Description:Displacement of [3H]RX821002 from human Alpha-2C adrenoceptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at human alpha2C ARMore data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:Agonist activity at human Alpha-2C adrenoceptor expressed in CHO cells assessed as induction of extracellular acidification by microphysiometryMore data for this Ligand-Target Pair