Found 11 Enz. Inhib. hit(s) with Target = 'Apelin receptor' and Ligand = 'BDBM50172371' 
Affinity DataKi: 0.370nMAssay Description:Displacement of [125I]-Apelin-13[Glp65, Nle75, Tyr77] from YFP epitope-tagged human APJ expressed in HEK-293 cells after 1 hr by gamma counting metho...More data for this Ligand-Target Pair
Affinity DataEC50: 16nMAssay Description:Induction of HA-tagged human APJ receptor internalization expressed in HEK-293 cells after 30 mins by ELISAMore data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at human APJ receptor expressed in HEK-293 cells assessed as dissociation of G-alpha-i1 protein after 5 mins by BRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.117nMAssay Description:Agonist activity at human APJ receptor by saphenous vein contraction assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Agonist activity at human APJ receptor assessed as Go activationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.70nMAssay Description:Agonist activity at human APJ receptor assessed as increase in beta-arrestin recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Induction of human APJ receptor internalization by cell based assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human APJ receptor assessed as Gi activationMore data for this Ligand-Target Pair
Affinity DataEC50: 69nMAssay Description:Agonist activity at human APJ receptor assessed as increase in beta-arrestin2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:Agonist activity at human APJ receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment after 30 mins by BRET assayMore data for this Ligand-Target Pair
Affinity DataEC50: 73nMAssay Description:Agonist activity at human APJ receptor assessed as increase in beta-arrestin1 recruitmentMore data for this Ligand-Target Pair
