Found 65 Enz. Inhib. hit(s) with Target = 'Beta-2 adrenergic receptor' and Ligand = 'BDBM25392' 
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]-(R,R')-methoxyfenoterol from human beta2 adrenergic receptor expressed in HEK cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 46nMAssay Description:Displacement of [3H]CGP12177 from human beta2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Tested for binding affinity against beta-2 adrenergic receptor in bovine lung using [3H]DHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 110nMAssay Description:Compound was evaluated for beta adrenergic binding affinity towards beta-2 receptor of bovine lungMore data for this Ligand-Target Pair
Affinity DataKi: 136nM ΔG°: -38.8kJ/molepH: 7.4 T: 2°CAssay Description:The displacement of [125I]-(-)iodopindolol binding from the beta2AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined...More data for this Ligand-Target Pair
Affinity DataKi: 192nMAssay Description:Displacement of [3H]-CGP-12177 from human beta2 adrenergic receptor expressed in HEK cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [3H]-DHA from recombinant human beta2 adrenoceptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 676nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. IC50, the mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Agonistic activity for Beta-2 adrenergic receptor was assessed by it's inhibitory effect on spontaneous contractions in isolated rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of spontaneous contractions in isolated rat uterusMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for its binding affinity towards beta-2 adrenergic receptor in rat soleus membrane by displacing(-)-isoproterenol (50 microM)More data for this Ligand-Target Pair
Affinity DataEC50: 58nMAssay Description:Agonistic activity (beta2- adrenergic) for the percent maximal relaxation of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataEC50: 0.160nMAssay Description:Activity at human beta-2 adrenergic receptor expressed in CHO cells by stimulation of cAMP productionChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human cloned beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation by beta-ga...More data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human recombinant beta2 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human beta2 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human recombinant beta2 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Agonist activity at recombinant human beta2 adrenoceptor expressed in HEK293T cells assessed as increase in IBMX-induced cAMP accumulation using [3H]...More data for this Ligand-Target Pair
Affinity DataEC50: 129nMAssay Description:Agonist activity at recombinant human beta2 adrenoceptor expressed in DU145 cells assessed as increase in cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human beta2 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonistic activity was assessed by measuring cAMP accumulation in CHO cell lines expressing cloned human Beta-2 adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human recombinant beta2 adrenergic receptor expressed in CHO cells assessed as induction of intracellular cAMP accumulation after...More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human cloned adrenergic beta2 receptor expressed in CHO cells assessed as increase in cAMP production after 2 days by radioimmuno...More data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:Binding affinity to human adrenergic beta2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 0.840nMAssay Description:Agonist activity at human recombinant adrenergic beta2 receptor expressed in CHO cells assessed as stimulation of cAMP level after 1 hr by enzyme imm...More data for this Ligand-Target Pair
Affinity DataEC50: 0.160nMAssay Description:Activity against human beta 2 adrenergic receptor (AR), expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as intracellular cAMP accumulation after 1 hrMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Agonist activity at human beta2 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring at basal tone assessed as bronchorelaxation activityMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at PK-tagged beta2 receptor (unknown origin) transfected in HEK293 cells after 90 mins by beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataEC50: 87nMAssay Description:Agonist activity at human beta2 receptor expressed in HEK293 cells cotransfected with Gqs5 protein assessed as [3H]IP3 accumulation after 120 mins by...More data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Agonist activity at guinea pig trachea beta2-adrenergic receptor assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
Affinity DataEC50: 31.6nMAssay Description:Agonist activity at beta2 adrenoceptor in guinea pig assessed as relaxation of histamine-induced tracheal ring contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Agonist activity at human cloned adrenergic beta2 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoassa...Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Agonist activity at human cloned adrenergic beta2 receptor expressed in CHO cells assessed as [125I]cAMP accumulation after 2 days by radioimmunoassa...Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKd: 309nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Agonist activity at recombinant human beta2 adrenergic receptor expressed in CHO cells assessed as accumulation of cyclic AMP after 30 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at human beta2-AR expressed in CHOK1 cells co-expressing Galpha15 measured after 21 secs to 120 secs by Calcium-4 dye based FLIPR as...More data for this Ligand-Target Pair
