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Found 5 Enz. Inhib. hit(s) with Target = 'Beta-2 adrenergic receptor' and Ligand = 'BDBM82498'
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  4.26nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  6.16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  6.60nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataKi:  8.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-2 adrenergic receptor(GUINEA PIG)
Ohio State University

Curated by PDSP Ki Database
LigandPNGBDBM82498(TMQ, 5,8-Difluoro)
Affinity DataEC50:  240nMAssay Description:Inhibitory activity against Beta-2 adrenergic receptor in guinea pig trachea after treatment with the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed