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Found 6 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50240563'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at dog beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at dog beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed