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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50264587'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50264587((R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamin...)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity at human cloned adrenergic beta3 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50264587((R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamin...)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at dog cloned adrenergic beta3 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed