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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50277509'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50277509(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-pyridin...)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50277509(3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-pyridin...)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed