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Found 3 Enz. Inhib. hit(s) with Target = 'Biotin--protein ligase' and Ligand = 'BDBM50039492'
TargetBiotin--protein ligase(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  182nMAssay Description:Inhibition of human recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataKi:  7.54E+5nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBiotin--protein ligase(Homo sapiens (Human))
University Of Adelaide

Curated by ChEMBL
LigandPNGBDBM50039492(CHEMBL1231498)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human recombinant HLCS using P67 as substrate after 2 hrs relative to vehicle-treated controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed