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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'CREB-binding protein' and Ligand = 'BDBM348901'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
CREB-binding protein


(Homo sapiens (Human))
BDBM348901
PNG
((4R)-4-methyl-6-[(E)-2- | US10206931, Example 3)
Show SMILES C[C@@H]1CC(=O)Nc2cccc(\C=C\c3ccncc3)c2N1
Show InChI InChI=1S/C17H17N3O/c1-12-11-16(21)20-15-4-2-3-14(17(15)19-12)6-5-13-7-9-18-10-8-13/h2-10,12,19H,11H2,1H3,(H,20,21)/b6-5+/t12-/m1/s1
PDB
MMDB

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KEGG

UniProtKB/SwissProt

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PC cid
PC sid
UniChem
US Patent
n/an/a 608n/an/an/an/an/an/a



Genentech Inc

US Patent


Assay Description
His/Flag epitope tagged CBP was cloned, expressed, and purified to homogeneity. CBP binding and inhibition was assessed by monitoring the engagement ...


US Patent US10206931 (2019)


BindingDB Entry DOI: 10.7270/Q2GM89FR
More data for this
Ligand-Target Pair