Affinity DataKi: 638nMAssay Description:Evaluated for binding affinity against recombinant human central cannabinoid receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 3.55E+7nMAssay Description:Displacement of [3H]CP-55940 from Cannabinoid receptor 1 of rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.61E+7nMAssay Description:Binding affinity at cannabinoid receptor 1 using rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.61E+7nMAssay Description:Cannabinoid receptor 1 binding affinity by measuring its ability to displace [3H]WIN-55212-2 in rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Concentration of compound required to inhibit 50% of [3H]-WIN- 55212 binding to Cannabinoid receptor 1 in rat cerebellum membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Binding affinity against brain Cannabinoid receptor 1 using [3H]-CP-55,940 as radioligand at 1.1 nM concentrationMore data for this Ligand-Target Pair