Affinity DataKi: 18.6nMAssay Description:Inhibition of [3H]-SR-141,716A binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 360nMAssay Description:Displacement of [3H]CP-55,940 binding to Cannabinoid receptor 1 in rat brain membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]-CP55940 from rat CB1 receptor by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Activity at human CB1 receptor by [35S]GTP-gamma-S binding stimulation assayMore data for this Ligand-Target Pair