Affinity DataKi: 748nMAssay Description:Ability to displace [3H]WIN-55212-2 radioligand from cannabinoid receptor 1 in rat cerebellar membraneMore data for this Ligand-Target Pair
Affinity DataKi: 829nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
Affinity DataKi: 856nMAssay Description:Ability to displace [3H]SR-141,716A radioligand from cannabinoid receptor 1 in rat cerebellar membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Inverse agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 690nMAssay Description:Inverse agonist activity at rat CB1 receptorMore data for this Ligand-Target Pair