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Found 5 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50147009'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
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Curated by ChEMBL
LigandPNGBDBM50147009(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-3-hexy...)
Affinity DataKi:  748nMAssay Description:Ability to displace [3H]WIN-55212-2 radioligand from cannabinoid receptor 1 in rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50147009(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-3-hexy...)
Affinity DataKi:  829nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50147009(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-3-hexy...)
Affinity DataKi:  856nMAssay Description:Ability to displace [3H]SR-141,716A radioligand from cannabinoid receptor 1 in rat cerebellar membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50147009(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-3-hexy...)
Affinity DataIC50:  631nMAssay Description:Inverse agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Instituto De Qu£Mica M£Dica

Curated by ChEMBL
LigandPNGBDBM50147009(5-(4-Chloro-phenyl)-1-(2,4-dichloro-phenyl)-3-hexy...)
Affinity DataIC50:  690nMAssay Description:Inverse agonist activity at rat CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed