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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50239215'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP55940 from human cloned CB1 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP 55940 from human CB1 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataEC50:  920nMAssay Description:Agonist activity at human cloned CB1 receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed