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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50384161'
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50384161(CHEMBL2029727)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50384161(CHEMBL2029727)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cells assessed as [35S]GTPgamma bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed