Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1R expressed in HEK293 cell membranes incubated for 90 mins by Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Antagonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as decrease in CP55940-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 1.62E+3nMAssay Description:Agonist activity at N-terminal Flag epitope tagged CB1 (unknown origin) expressed in HTLA cells assessed as increase of beta-arrestin recruitment by ...More data for this Ligand-Target Pair