Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50067498'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CP-55940 from human CB2 receptor expressed in COS cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-CP55940 from rat CB2 receptor by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50067498((6aS,10aS)-3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl...)
Affinity DataEC50:  0.251nMAssay Description:Agonist activity at human CB2 receptor transfected in CHO cells by [35]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed