Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Cathepsin K' and Ligand = 'BDBM50138842'
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50138842(2,4-dimethylpentan-3-yl(S)-1,2-dioxo-1-((R)-1-phen...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory activity against human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50138842(2,4-dimethylpentan-3-yl(S)-1,2-dioxo-1-((R)-1-phen...)
Affinity DataIC50:  2.51nMAssay Description:Inhibition of human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50138842(2,4-dimethylpentan-3-yl(S)-1,2-dioxo-1-((R)-1-phen...)
Affinity DataIC50:  2.54nMAssay Description:Concentration required to inhibit 50% of cysteine protease cathepsin K of humanMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50138842(2,4-dimethylpentan-3-yl(S)-1,2-dioxo-1-((R)-1-phen...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity of the compound against rat cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50138842(2,4-dimethylpentan-3-yl(S)-1,2-dioxo-1-((R)-1-phen...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory concentration against recombinant human cathepsin KMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed