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Found 2 Enz. Inhib. hit(s) with Target = 'Coagulation factor X' and Ligand = 'BDBM294042'
TargetCoagulation factor X(Homo sapiens (Human))
North China Pharmaceutical New Drug R&D

US Patent
LigandPNGBDBM294042(US10106557, Compound 8)
Affinity DataKi:  1.92nMpH: 8.3Assay Description:The inhibitory activity on coagulation factor Xa activity in human was measured by using Tris-HCl buffer (50 mM, pH 8.3, 150 mM NaCl). A buffer of 50...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor X(Rattus norvegicus (rat))
North China Pharmaceutical New Drug R&D

US Patent
LigandPNGBDBM294042(US10106557, Compound 8)
Affinity DataKi:  3.17nMpH: 8.3Assay Description:The inhibitory activity on coagulation factor Xa activity in rats was measured by using Tris-HCl buffer (50 mM, pH 8.3, 150 mM NaCl). A buffer of 50 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent