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Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2' and Ligand = 'BDBM7157'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute Of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7157(3-Phenylacetamidoaminopyrazole deriv. 34 | CHEMBL1...)
Affinity DataIC50:  67nMAssay Description:Inhibition of CDK2/Cyclin A (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute Of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7157(3-Phenylacetamidoaminopyrazole deriv. 34 | CHEMBL1...)
Affinity DataKd:  6.89E+3nMpH: 7.5 T: 2°CAssay Description:ThermofluorMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Institute Of Chemical Biology (Csir)

Curated by ChEMBL
LigandPNGBDBM7157(3-Phenylacetamidoaminopyrazole deriv. 34 | CHEMBL1...)
Affinity DataKd:  5.83E+4nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair