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Found 8 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 2' and Ligand = 'BDBM8065'
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKd:  2.59E+3nMpH: 7.5 T: 2°CAssay Description:ThermofluorMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKd:  557nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKd:  161nMAssay Description:OctetRed_Method2More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKon:  0.0367M-1s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKon:  0.0200M-1s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKd:  557nMAssay Description:OctetRed_Method1More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKoff:  1.13E+5s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Csar

LigandPNGBDBM8065(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 36 | 3...)
Affinity DataKoff:  1.58E+5s-1Assay Description:OctetRed_Method3More data for this Ligand-Target Pair
In DepthDetails PubMed