TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 6.17nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Displacement of [3H]SCH23390 from porcine striatal membranes D1 receptor by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Affinity for Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards Dopamine receptor D1More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]SCH233930 from human D1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:Ability to displace [3H]-SCH- 23390 (0.2 nM) from corpus striatum of rat Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity was measured against dopamine receptor D1 in rat using [3H]SCH-23390 as radioligandMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Compound was tested for the binding affinity against human cloned Dopamine receptor D1 by radioligand ([3H]-SCH-23390) binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 71nMAssay Description:Binding Affinity was determined against Dopamine receptor D1 in rat striatal membranes using [3H]- SCH 23390 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:In vitro binding affinity against Dopamine receptor D1 in rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:Binding affinity against dopamine receptor D1More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Binding affinity for human recombinant dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Displacement of [3H]SCH 23390 from pig dopamine D1 receptor in striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Displacement of [3H]SCH23390 from D1 receptor from porcine cerebral cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Compound was evaluated for its affinity (pKi) to inhibit [3H]SCH-23390 binding to the Dopamine receptor D1Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Inhibition constant for in vitro inhibition of [3H]-SCH- 23390 binding to striatal membranes Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in pig striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 rat striatal membraneMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 107nMAssay Description:Inhibition of human dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity to human cloned dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Binding affinity measured at the Dopamine receptor D1 by the inhibition of [3H]-SCH-23,390 binding to rat striatum using unlabeled apomorphine for no...More data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:In vitro ability to displace [3H]SCH-23390 binding from Dopamine 1 (D1) receptor in rat striatal membrane.More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Universidad De Santiago De Compostela
Curated by ChEMBL
Universidad De Santiago De Compostela
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Binding affinity towards human Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 318nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in CRL:CD(SD)BR-COBS rat striatum by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataKi: 318nMAssay Description:Binding affinity to dopamine D1 receptor in rat striatum by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 318nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to rat dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 318nMAssay Description:Half-maximal inhibition of [3H]-SCH- 23390 binding to Dopamine receptor D1 in rat striatal homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 318nMAssay Description:In vitro binding affinity towards Dopamine receptor D1 in rat tissue homogenate using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 359nMAssay Description:Inhibition of [3H]-SCH-23,390 binding to rat Dopamine receptor D1More data for this Ligand-Target Pair
Affinity DataKi: 467nMAssay Description:Tested for binding affinity towards rat striatal dopamine receptor D1 using [3H]-SCH- 23390 as radioligandMore data for this Ligand-Target Pair