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Found 3 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50378001'
TargetD(3) dopamine receptor(Homo sapiens (Human))
The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services

US Patent
LigandPNGBDBM50378001(CHEMBL1627321 | US8748608, 36)
Affinity DataKi:  0.260nMAssay Description:Methods for performing in vitro dopamine receptor binding studies are described in Huang et al. J. Med. Chem. 44:1815-1826 (2001) and Luedtke et al. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services

US Patent
LigandPNGBDBM50378001(CHEMBL1627321 | US8748608, 36)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125]IABN from human D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services

US Patent
LigandPNGBDBM50378001(CHEMBL1627321 | US8748608, 36)
Affinity DataIC50:  25.7nMAssay Description:Antagonist activity at human D3 receptor expressed in HEK293 cells assessed as inhibition of quinpirole-stimulated mitogenesisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed