Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellumMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
R. W. Johnson Pharmaceutical Research Institute
Curated by PDSP Ki Database
R. W. Johnson Pharmaceutical Research Institute
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: >1.20E+4nMAssay Description:Displacement of [3H]DADLE from human recombinant delta opioid receptor expressed in CHO cell membranes after 2 hrs by liquid scintillation counting a...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKi: 1.25E+4nMAssay Description:Displacement of [3H]DADLE from human delta opioid receptor expressed in CHO cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of [125I]-(D-Pro10)-Dynorphin A binding to human kappa opioid receptor from membranes of HEK293 cellsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataIC50: 5.84E+3nMAssay Description:Binding affinity towards Opioid receptor mu 1 by the displacement of [125I]Enkephalin; Not determinedMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKd: 1.98E+3nMAssay Description:Binding affinity against Mu opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes in unblocked conditionMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Pennsylvania
Curated by PDSP Ki Database
University Of Pennsylvania
Curated by PDSP Ki Database
Affinity DataKd: 1.98E+3nMAssay Description:Binding affinity against kappa opioid receptor using [35S]GTP-gamma-S, binding assay in guinea pig caudate membranes blocked with 6 nM nor-BNIMore data for this Ligand-Target Pair