Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of [3H]-naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 2.65E+3nMAssay Description:Displacement of [3H]Ile5,6-deltorphin II from opioid receptor delta 1 of rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 3.39E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor (unknown origin) expressed in CHO cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataKi: 3.94E+3nMAssay Description:Binding affinity towards delta receptor in rat brain using [3H]DSLETMore data for this Ligand-Target Pair
Affinity DataKi: 5.65E+3nMAssay Description:Displacement of [3H]Ile5,6deltorphin-2 from delta opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 6.08E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in rat brain P2 synaptosomeMore data for this Ligand-Target Pair
Affinity DataKi: 6.09E+3nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 6.09E+3nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.42E+3nMAssay Description:Displacement of [3H]DPDPE from Myc-tagged delta opioid receptor expressed in HEK293 cells after 60 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Displacement of [3H]DPDPE from rat cortex delta opioid receptor after 2.5 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 7.90E+3nMAssay Description:Displacement of [3H]deltrophin-2 from human recombinant DOR expressed in CHO cell membranes incubated for 2 hrs by liquid scintillation counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 8.36E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 8.36E+3nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Wistar rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 8.50E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Wistar rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 8.77E+3nMAssay Description:Displacement of [3H]DPDPE from DOR in Wistar rat brain membranes measured after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 8.77E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin2 from delta opioid receptor in rat brain membrane homogenate by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 9.23E+3nMAssay Description:Binding affinity against rat brain opioid receptor delta 1 using [3H]-DPDPE radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 9.23E+3nMAssay Description:Displacement of [3H]-[Ile5,6]-deltorphin-2 from Wistar rat brain membrane DOPMore data for this Ligand-Target Pair
Affinity DataKi: 9.62E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin-2 from DOR in Wistar rat brain homogenates by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-DPDPE from Wistar rat delta opioid receptor incubated for 3 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]Ile5,6deltorphin-2 from delta opioid receptor in Wistar rat brain membranes by liquid scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 15nMAssay Description:Agonist activity at delta opioid receptor by inhibition of electrically evoked muscle contraction in isolated mouse vas deferensMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 22nMAssay Description:Agonist activity at delta opioid receptor in Kunming mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 25.8nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 48.2nMAssay Description:In vitro inhibitory concentration against Opioid receptor delta 1 was measured using mouse vas deferens assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 344nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 344nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked muscle contractionsMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 510nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically evoked contractionMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 510nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin-2 from delta opioid receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin 2 from delta opioid receptor in Wistar rat brain membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin-2 from DOR in Wistar rat brain membranes by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H][Ile5,6]deltorphin-2 from delta opioid receptor in Wistar rat brain membranes after 120 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [3H](Ile5,6)deltorphin-2 from DOR in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]naltrindole from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+4nMAssay Description:Displacement of [3H]deltorphin2 from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(MOUSE)
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Clinical Research Institute Of Montreal
Curated by PDSP Ki Database
Affinity DataIC50: 5.10E+5nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deference assessed as inhibition of electrically-stimulated contractionMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Activity at delta opioid receptor assessed as increase in calcium level in CHO cells by aequorin luminescence based calcium assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at delta opioid receptor expressed in CHO cells assessed as release of intracellular calcium ions by aequorin luminescence-based ...More data for this Ligand-Target Pair