Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Dual specificity mitogen-activated protein kinase kinase 1' and Ligand = 'BDBM25117'
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Ambit Biosciences

Curated by ChEMBL
LigandPNGBDBM25117(AG-013736 | AXITINIB | N-methyl-2-({3-[(E)-2-(pyri...)
Affinity DataKd:  2.70E+3nMAssay Description:Binding constant for MEK1 kinase domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed