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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Dual-specificity tyrosine-phosphorylation regulated kinase 1A' and Ligand = 'BDBM50187066'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Dual-specificity tyrosine-phosphorylation regulated kinase 1A


(Mus musculus)
BDBM50187066
PNG
(4-(4-hydroxy-3-methoxybenzylidene)-1-(3-chlorophen...)
Show SMILES COc1cc(C=C2C(=O)NN(C2=O)c2cccc(Cl)c2)ccc1O
Show InChI InChI=1S/C17H13ClN2O4/c1-24-15-8-10(5-6-14(15)21)7-13-16(22)19-20(17(13)23)12-4-2-3-11(18)9-12/h2-9,21H,1H3,(H,19,22)
PDB
MMDB

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PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a>5.00E+4n/an/an/an/an/an/a



Research Center IDRTech Inc.

Curated by ChEMBL


Assay Description
Inhibition of mouse Dyrk1A autophosphorylation in HEk293 cells


Bioorg Med Chem Lett 16: 3772-6 (2006)


Article DOI: 10.1016/j.bmcl.2006.04.042
BindingDB Entry DOI: 10.7270/Q2K938BX
More data for this
Ligand-Target Pair