Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Endothelin-1 receptor' and Ligand = 'BDBM50045227'
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50045227((S)-3-[2-((R)-2-Acetylamino-3-phenyl-propionylamin...)
Affinity DataIC50:  750nMAssay Description:Displacement of [125I]-ET-1 from Endothelin A receptor of rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin-1 receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50045227((S)-3-[2-((R)-2-Acetylamino-3-phenyl-propionylamin...)
Affinity DataIC50:  2.45E+3nMAssay Description:Binding affinity against ET A receptor from rabbit renal artery vascular smooth muscle cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed