Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor' and Ligand = 'BDBM202376'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research

US Patent
LigandPNGBDBM202376(US10081606, Compound I-8 | US9238629, I-8 | US9765...)
Affinity DataIC50:  65nMpH: 7.5 T: 2°CAssay Description:Briefly, 10x stocks of EGFR-WT (PV3872) from Invitrogen and EGFR-T790M/L858R (40350) from BPS Bioscience, San Diego, Calif., 1.13x ATP (AS001A) and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research

US Patent
LigandPNGBDBM202376(US10081606, Compound I-8 | US9238629, I-8 | US9765...)
Affinity DataIC50:  65nMpH: 7.5Assay Description:The mechanics of the assay platform are best described by the vendor (Invitrogen, Carlsbad, Calif.) on their web site at the following URL: www.invit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research

US Patent
LigandPNGBDBM202376(US10081606, Compound I-8 | US9238629, I-8 | US9765...)
Affinity DataIC50:  65nMAssay Description:The mechanics of the assay platform are best described by the vendor (Invitrogen, Carlsbad, Calif.) on their web site at the following URL: www.invit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research

US Patent
LigandPNGBDBM202376(US10081606, Compound I-8 | US9238629, I-8 | US9765...)
Affinity DataEC50: >1.00E+3nMAssay Description:The mechanics of the assay platform are best described by the vendor (Invitrogen, Carlsbad, Calif.) on their web site at the following URL: www.invit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Celgene Avilomics Research

US Patent
LigandPNGBDBM202376(US10081606, Compound I-8 | US9238629, I-8 | US9765...)
Affinity DataEC50: >1.00E+3nMAssay Description:To assess phosphor-EGFR signaling, blots were probed with rabbit anti-Phospho-EGFR (Y1068) and mouse total anti-EGFR antibodies. Phospho-EGFR signal ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent