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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Formyl peptide receptor 2' and Ligand = 'BDBM50559840'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Formyl peptide receptor 2


(Mus musculus)
BDBM50559840
PNG
(CHEMBL4760897)
Show SMILES COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(Cl)s2)c(F)c1
Show InChI InChI=1S/C16H14ClF2N3O3S/c1-25-7-4-9(18)13(10(19)5-7)8-6-20-15(23)14(8)22-16(24)21-12-3-2-11(17)26-12/h2-5,8,14H,6H2,1H3,(H,20,23)(H2,21,22,24)/t8-,14-/m0/s1
KEGG

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
PubMed
n/an/an/an/a 1.40n/an/an/an/a



Kyorin Pharmaceutical Co. Ltd.

Curated by ChEMBL


Assay Description
Agonist activity at mouse FPR2 expressed in HEK 293 cells co-expressing Galpha15 measured every 1.5 sec for 80 sec by Fluo-4 NW staining based scanni...


J Med Chem 63: 9003-9019 (2020)

More data for this
Ligand-Target Pair