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Found 2 Enz. Inhib. hit(s) with Target = 'G-protein coupled estrogen receptor 1' and Ligand = 'BDBM349623'
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349623((4-fluoro-2,6-dimethylphenyl)(3-(4-(2- (3-(fluorom...)
Affinity DataIC50: <1.00E+3nMAssay Description:All reagents used in this assay was supplied in the Human ERα Reporter Assay by Indigo Biosciences # IB00401. In an effort to screen selective e...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled estrogen receptor 1(Homo sapiens (Human))
G1 Therapeutics

US Patent
LigandPNGBDBM349623((4-fluoro-2,6-dimethylphenyl)(3-(4-(2- (3-(fluorom...)
Affinity DataIC50: <1.00E+3nMAssay Description:A screening strategy was implemented utilizing an In-Cell Western assay to measure their ability to degrade the estrogen receptor in vitro. MCF7 cell...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent