TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Janssen Research Foundation
Curated by PDSP Ki Database
Janssen Research Foundation
Curated by PDSP Ki Database
Affinity DataKi: 5.30nMAssay Description:Binding affinity towards human histamine H1 receptorMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Janssen Research Foundation
Curated by PDSP Ki Database
Janssen Research Foundation
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Displacement of [3H]pyrilamine from histaminergic H1 receptor guinea pig cerebellumMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity to human cloned histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity to H1 histamine receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Binding affinity towards human H1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Displacement of [3H]mepyramine from H1R in rat brainMore data for this Ligand-Target Pair