TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Queen'S Medical Centre
Curated by PDSP Ki Database
Queen'S Medical Centre
Curated by PDSP Ki Database
Affinity DataKi: 7.94E+4nMAssay Description:Displacement of [3H]mepyramine from human wild-type histamine H1 receptor expressed in COS-7 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibitory activity against human Histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 191nMAssay Description:Agonist activity at human H1 receptor expressed in insect Sf9 cells co-expressing RGS4 assessed as gamma[32P]GTP binding by liquid scintillation coun...More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Inhibition of human Histamine H1 receptor using [3H]-pyrilamineMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity at human H1 receptor expressed in 293-EBNA cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 190nMAssay Description:Activity at human recombinant histamine H1 receptor expressed in Sf9 cells coexpressing RGS4 by steady-state GTPase activity assayMore data for this Ligand-Target Pair
Affinity DataEC50: 191nMAssay Description:Agonist activity at human histamine H1 receptor expressed in Sf9 cells coexpressing RGS4 by steady-state GTPase assayMore data for this Ligand-Target Pair
Affinity DataEC50: 191nMAssay Description:Activity at human recombinant histamine H1 receptor expressed in Sf9 cells coexpressing RGS4 by steady-state GTPase activity assayMore data for this Ligand-Target Pair